Enantioselective α-Aminophosphonate Functionalization of Indole Ring through an Organocatalyzed Friedel-Crafts Reaction
The Journal of Organic Chemistry 84(2) : 1094-1102 (2018)
Laburpena
Chiral phosphoric acids efficiently catalyze the asymmetric
Friedel−Crafts reaction of several indoles with α-iminophosphonates
to afford enantioenriched hybrid α-aminophosphonate
functionalized indole derivatives.